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Creative PeptidesModel 514814-49-4 - PMX 205

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Potent C5a receptor peptide antagonist (IC50 = 31 nM). Ameliorates experimentally-induced colon inflammation in mice. Reduces fibrillar amyloid deposits, decreases hyperphosphorylated tau levels and rescues cognitive function in a mouse model of Alzheimer's Disease. Orally active and brain penetrant.http://www.creative-peptides.com/product/pmx-item-10-101-154-33641.html